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β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Letswai CAS:24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Letswaike coenzyme e ajoang haholo linthong tse phelang, E nka karolo liketsong tsa ho fokotsa oxidation. E sebetsa e le mojari oa lielektrone liketsong tse 'maloa, e fetoloa ka mokhoa o fapaneng (NADP+) le ho fokotsoa (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Letswaike ntho eo nicotinic acid amide adenine dinucleotide le molek'hule ea phosphate li tlamiloeng ka tlamo ea ester. Ke receptor ea haedrojene 'me e ka sebelisoa bakeng sa nts'etsopele le nts'etsopele ea mefuta e fapaneng ea li-reagent tsa tlhahlobo ea in vitro.
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β-Nicotinamide Adenine Dinucleotide Letsoai la Lithium (NAD Lithium letsoai) CAS:64417-72-7
β-Nicotinamide Adenine Dinucleotide Letswai la lithiumke coenzyme e bohareng ba metabolism. E fumaneha liseleng tsohle tse phelang, NAD e bitsoa dinucleotide hobane e na le li-nucleotide tse peli tse kopantsoeng ka lihlopha tsa tsona tsa phosphate. Nucleotide e 'ngoe e na le adenine nucleobase le nicotinamide e 'ngoe. NAD e teng ka mefuta e 'meli: sebopeho se nang le oxidized le se fokolitsoeng, se khutsufalitsoeng e le NAD+ le NADH (H bakeng sa haeterojene), ka ho latellana.
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Venlafaxine CAS:93413-69-5
Venlafaxine ke moriana o thibelang ho tepella maikutlo oa sehlopha sa serotonin le norepinephrine reuptake inhibitor (SNRI). Moriana ona o qalile ho hlahisoa ke Wyeth ho 19Chemicalbook93 'me joale o rekisoa ke Pfizer. Moriana ona o amohetsoe bakeng sa kalafo ea lefu la khatello ea maikutlo le leholo (MDD), lefu la ho tšoenyeha ka kakaretso (GAD), le khatello ea maikutlo e amanang le ho tšoenyeha.
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Ciclopirox Ethanolamine CAS:41621-49-2 Mofani oa Moetsi
Ciclopirox ethanolamine ke setlhare se seholo se loantšang li-fungus, hape se na le ts'ebetso ea antibacterial khahlanong le libaktheria tse ngata tsa Gram-positive le Gram-negative, 'me se na le thepa ea ho thibela ho ruruha. E sebelisoa e le kalafo ea letlalo la fungus le tšoaetso ea manala.
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Desvenlafaxine Succinate CAS:386750-22-7
Desvenlafaxine Succinate ke serotonin e habeli le norepinephrine reuptake inhibitor (SNRI) e ileng ya amohelwa bakeng sa kalafo ya lefu la kgatello e kgolo ya maikutlo (MDD) United States ka 2008. E le ho ntlafatsa katleho le polokeho ya venlafaxine, Wyeth o ile a sibolla mme a ntshetsa pele e nngwe ya di-metabolite tse kgolo tsa venlafaxine, e leng O-desmethyl metabolite (desvenlafaxine).
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Doxazosin Mesylate CAS: 77883-43-3 Mofani oa Moetsi
Doxazosin mesylate ke motsoako oa quinazoline o thibelang ho sebelisoa ha mofuta oa alpha1 oa li-receptor tsa alpha adrenergic. Doxazosin mesylate ke moloko o mocha oa quinazolone α1 receptor blocker e ntlafalitsoeng ke k'hamphani ea Pfizer (United States), E na le halofo ea bophelo bo bolelele, e sebelisa litlamorao tsa eona tsa ho atolosa methapo ea mali, ho fokotsa ho hanyetsa methapo ea mali le ho theola khatello ea mali ka ho thibela receptor ea a1. E khothalelitsoe kantle ho naha e le meriana ea pele ea bongaka ea ho thibela khatello e phahameng ea mali le kalafo ea lefu la prostate.
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L-Isoleucine CAS: 73-32-5 Mofani oa Moetsi
L-Isoleucine, e tsejoang hape e le Isoleucine, ke amino acid e leng isomer ea leucine. E bohlokoa ho etseng hemoglobin le ho laola maemo a tsoekere le matla maling. L-Isoleucine ke isomer ea L-leucine 'me ke amino acid ea bohlokoa. E entsoe ho tsoa ho threonine 'me ke amino acid ea hydrophobic ea chain e nang le makala.
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Captopril CAS: 62571-86-2 Mofani oa Moetsi
Captopril ke e 'ngoe ea li-inhibitor tsa angiotensin-converting enzyme tse ithutoang ka ho fetisisa tse hlahisoang e le moriana o fokotsang khatello ea mali. E thibela enzyme e fetolang angiotensin, e thibelang ho thehoa ha angiotensin II le ho imolla phello ea eona ea ho koala methapo ea mali le ea mali. Khatello e akaretsang ea methapo ea mali e ea fokotseha, e leng se fellang ka ho fokotseha ha khatello ea mali.
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Candesartan CAS:139481-59-7 Mofani oa Moetsi
Candesartan ke mohanyetsi oa angiotensin II receptor I (AT1), IC50s=1.12 le 2.86 nM bakeng sa cortex ea adrenal ea likhomo le aorta ea mmutla ka ho latellana. E thibela ka khetho ho honyela ho bakoang ke angiotensin II ha meqolo ea aortic ea mmutla ka mokhoa o sa amaneng le ho honyela ho bakoang ke metsoako e meng e kang norepinephrine, KCl, serotonin, PGF2α kapa endothelin.
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Candesartana Cilexetila CAS:145040-37-5
Candesartan Celexetil ke analoge ea ester ea mohanyetsi oa angiotensin II Candesartan (sc-217825). Khahlano ea receptor ena e thibela ho tlama ha angiotensin II, vasoconstrictor e matla. Sena se na le phello e akaretsang ea ho ruruha ha methapo ea mali le keketseho ea molumo oa mali oa capillary. Candesartan Celexetil Ester ke thibelo ea AT1.
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Bupropion CAS:34911-55-2 Mofani oa Moetsi
Bupropion ke ketone e nkhang hamonate e leng propiophenone e jereng sehlopha sa tert-butylamino boemong ba 2 le sebaka sa chloro boemong ba 3 hodima lesale la phenyl. E na le karolo e le moriana o thibelang ho tepella maikutlo, o silafatsang tikoloho le o bakang xenobiotic. Ke motsoako oa bobeli oa amino, setho sa monochlorobenzenes le ketone e nkhang hamonate.
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Bezafibrate CAS:41859-67-0 Mofani oa Moetsi
Bezafibrate ke amide ea monocarboxylic acid e fumanoang ka ho kopana ha sehlopha sa carboxy sa 4-chlorobenzoic acid le sehlopha sa amino sa 2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic acid. Benafibrate e sebelisetsoa ho phekola hyperlipidaemia. E na le karolo e le xenobiotic, e silafatsang tikoloho, e sireletsang gero le moriana o thibelang li-lipidemic. Ke monocarboxylic acid, aromatic ether, setho sa monochlorobenzenes le monocarboxylic acid amide. E amana ka mokhoa o sebetsang le propionic acid.
