Lebanta le Tsela: Tšebelisano-'moho, Kutloano le ho Hlōla ka Botlalo
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Venlafaxine CAS:93413-69-5

Venlafaxine ke moriana o thibelang ho tepella maikutlo oa sehlopha sa serotonin le norepinephrine reuptake inhibitor (SNRI). Moriana ona o qalile ho hlahisoa ke Wyeth ho 19Chemicalbook93 'me joale o rekisoa ke Pfizer. Moriana ona o amohetsoe bakeng sa kalafo ea lefu la khatello ea maikutlo le leholo (MDD), lefu la ho tšoenyeha ka kakaretso (GAD), le khatello ea maikutlo e amanang le ho tšoenyeha.


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Venlafaxine e ka thibela ho nkuwa hape ha NA le 5-HT, mme ya boela ya thibela hanyane ho nkuwa hape ha dopamine. Thibelo ya in vitro ya di-receptor tsa cholinergic, di-receptor tsa histamine α Di-receptor ka bobedi ha di na kamano. Ho monywa ha mala ho hotle, mme Chemicalbook e tshediswa ke cytochrome P45011D6 sebeteng mme e ntshwa ke moroto. T1/2 ya di-metabolite tse kgolo tse sebetsang e tloha dihoreng tse 5 ho isa ho tse 11. Kamora dibeke tse 3, mahloriso a tsitsitseng a fihlelletswe. E sebedisetswa kalafo ya kgatello ya maikutlo.

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Tlhahisoleseling e 'Ngoe:

Sebopeho C17H27NO2
Teko 99%
Ponahalo Phofo e tšoeu ea kristale
Nomoro ea CAS 93413-69-5
Ho paka 25KG
Bophelo ba Shelofo lilemo tse 2
Polokelo Boloka sebakeng se pholileng le se omileng
Setifikeiti ISO.

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