Lebanta le Tsela: Tšebelisano-'moho, Kutloano le ho Hlōla ka Botlalo
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Olmesartan Medoxomil CAS:144689-63-4 Mofani oa Moetsi

Olmesartan Medoxomil, ke mohanyetsi e mocha oa receptor ea angiotensin II ea mofuta oa 1 ea kgetho le ea tlholisano 'me o thibela ka matla likarabelo tsa khatello e bakoang ke Ang.ll. Sethethefatsi sena se thibetse ka tlholisano ho tlamahana ha [125I1]-All ho li-receptor tsa AT1 ka har'a li-membrane tsa adrenal cortical tsa likhomo, empa ha se na phello ho tlamahaneng le li-receptor tsa AT2 ka har'a li-membrane tsa cerebellar tsa likhomo. Olmesartan medoxomil e boetse e bontšitsoe e fokotsa khatello ea mali haholo ka katleho ho feta losartan le captopril ea ACE inhibitor le ka katleho joalo ka pbloker atenolol.


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Tšebeliso le Phello

Olmesartan medoxomil ke mohanyetsi oa angiotensin II receptor o sebelisetsoang ho phekola khatello e phahameng ea mali. Olmesartan e sebetsa ka ho thibela ho tlama ha angiotensin II ho li-receptor tsa AT1 ka har'a mesifa ea methapo ea mali. Ka ho thibela ho tlama ho e-na le ho kopanya angiotensin II, olmesartan e thibela karabelo e mpe ea taolo mabapi le ho ntšoa ha renin. Olmesartan medoxomil ke moriana o tšehetsang ho tlosoa ha metabolite e sebetsang, olmesartan. Olmesartan e na le mokhoa o habeli oa ho ntša, ka hoo e ka bang 60% e tlosoa ke sebete 'me e setseng e tlosoa ke liphio. Maemong a ho se sebetse hantle ha liphio kapa sebete, tsela e 'ngoe ea ho ntša e ka lefella e senyehileng.

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Tlhahisoleseling e 'Ngoe:

Sebopeho C29H30N6O6
Teko 99%
Ponahalo Phofo e tšoeu ho isa ho beige
Nomoro ea CAS 144689-63-4
Ho paka 25KG
Bophelo ba Shelofo lilemo tse 2
Polokelo Boloka sebakeng se pholileng le se omileng
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