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Celecoxib CAS:169590-42-5 Mofani oa Moetsi
Celecoxib ke setho sa sehlopha sa pyrazoles e leng 1H-pyrazole e nkeloang sebaka maemong a 1, 3 le 5 ke lihlopha tsa 4-sulfamoylphenyl, trifluoromethyl le p-tolyl, ka ho latellana. Ke sethibela-cyclooxygenase-2, e sebelisoa kalafong ea ramatiki. E na le karolo e le sethibela-cyclooxygenase 2, sethibela-geroprotector, sethethefatsi se seng sa steroidal se thibelang ho ruruha le setlhare se kokobetsang bohloko se seng sa lithethefatsi. Ke setho sa toluene, sulfonamide, setho sa pyrazoles le motsoako oa organofluorine.
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Palmitoylethanolamide CAS: 544-31-0 Mofani oa Moetsi
Palmitoylethanolamide (PEA) ke amide e mafura e hlahisoang 'meleng e tlamang le ho kenya tšebetsong peroxisome proliferator-activated receptor alpha (PPAR-α). Qalong e ne e hlalosoa e le agonist ho receptor ea cannabinoid ea mofuta oa 2 (CB2), leha joale ho lemohuoa hore PEA ha e tlame ho li-receptor tsa cannabinoid. PEA e tsejoa e na le thepa ea ho thibela ho ruruha, ho kokobetsa bohloko le ho sireletsa methapo ea kutlo. Litlatsetso tsa PEA li 'nile tsa sebelisoa ke batho ba nang le bohloko bo sa foleng hammoho le ba nang le bohloko ba neuropathic.
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N-Acetyl-L-Carnitine HCl CAS: Mofani oa Moetsi oa 5080-50-2
Acetyl-L-carnitine ke mofuta oa acetyl oa L-carnitine ea bohlokoa ea mitochondrial metabolite e fetoloang ke li-esterase tsa plasma ho ba carnitine. Acetyl-L-carnitine e thusa ho monya acetyl-CoA ho ba mitochondria nakong ea oxidation ea mafura a acid, e ntlafatsa tlhahiso ea acetylcholine, 'me e hlohlelletsa tlhahiso ea protheine le membrane phospholipid. Bophelong, acetyl-L-carnitine (100 mg/kg) e eketsa maemo a protheine ea receptor ea mGlu2/3 le meeli ea bohloko ba mechini mohlaleng oa toeba oa bohloko bo sa foleng ba ho ruruha bo bakoang ke adjuvant e felletseng ea Freund.
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Esomeprazole Magnesium CAS:161973-10-0
Esomeprazole Magnesium, proton-pump inhibitor (PPI), ke S-isomer ea omeprazole. Esomeprazole e na le leiboleng le amohetsoeng ke FDA bakeng sa ho sebelisoa kalafong ea lefu la reflux la gastroesophageal (GERD) le nang le matšoao, ho kenyeletsoa le pholiso le tlhokomelo ea pholiso ea esophagitis e senyehileng le e le karolo ea mokhoa oa meriana e meraro bakeng sa tšoaetso ea Helicobacter pylori.
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Asiti ea ribonucleic e tsoang tomosong ea moapehi CAS: 63231-63-0
Ribonucleic acid (RNA) ke sesebelisoa se etsang filimi holim'a metsi se nang le ts'ebetso ea mongobo. Ena ke polyribonucleotide e fumanoang khubung le cytoplasmeng ea lisele. Phetisetso ea RNA e arotsoe ho tomoso ea biri. Phetisetso ena ea RNA e ikhethile bakeng sa phetisetso ea amino acid phenylalanine.
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Cystine CAS: 923-32-0 Mofani oa Moetsi
Cystine e thusa ho theheng letlalo 'me e bohlokoa bakeng sa ho ntša chefo 'meleng. Ka ho fokotsa bokhoni ba 'mele ba ho monya koporo, cystine e sireletsa lisele chefong ea koporo. Ha e se e fetotsoe, e tla ntša sulfuric acid, 'me sulfuric acid e tla sebelisana ka lik'hemik'hale le lintho tse ling ho eketsa ts'ebetso ea ho ntša chefo 'meleng oa tsamaiso eohle ea metabolism.
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L-Arginine L-Glutamate CAS:4320-30-3 Mofani oa Moetsi
L-Arginine L-Glutamateke mofani oa naetrojene bakeng sa tlhahiso ea nitric oxide.L-Arginine L-Glutamatee ka sebelisoa bakeng sa hypofunction e kaholimo ea mala kapa ho se sebetse hantle joalo ka lipatlisiso tsa dyspepsia ea ts'ebetso.
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Coenzyme A sodium salt hydrate CAS:55672-92-9
Coenzyme A e nang le letsoai la sodium hydrateke karolo ea bohlokoa ea cofactor litsamaisong tse phelang 'me e hlahisoa ho tsoa ho pantothenic acid (vithamine B5). Maemo a CoA ho mitochondria le peroxisomes a tsamaellana le 2-5 mM le 0.7 mM, ka ho latellana.Coenzyme A e nang le letsoai la sodium hydrateke coenzyme e nolofalletsang karabelo ea phetisetso ea li-enzyme tsa acyl-group le ho tšehetsa tlhahiso le oxidation ea mafura a acid.
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Indometacin CAS: 53-86-1 Mofani oa Moetsi
Indomethacin (Indocin) e sebelisoa kalafong ea ramatiki e matla ea gouty, ramatiki ea rheumatoid, ankylosing spondylitis, le osteoarthritis. Ha e khothalletsoe ho sebelisoa e le moriana o bonolo oa ho kokobetsa bohloko kapa oa ho fokotsa ho ruruha ka lebaka la bokhoni ba eona ba chefo. Indomethacin e sebelisoa ho ramatiki ea rheumatoid, polyarthritis e tšoaetsanoang e sa tobang, ramatiki ea gouty, osteoarthritis, ankylosing spondylitis, arthrosis, bohloko ba mokokotlo, neuralgia, myalgia, le mafu a mang a tsamaeang le ho ruruha.
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Tetraethylene Glycol CAS: 112-60-7 Mofani oa Moetsi
Tetraethylene glycol ke polymer e nang le diyuniti tsa ethylene glycol monomer le dihlopha tse pedi tsa terminal hydroxyl. Dihlopha tsa hydroxyl di ka arabela ho ntsha motsoako ona ho ya pele. Dikomporo tsa ethylene glycol di na le dibopeho tse tshabang metsi. Ho qhibiliha ha polymer ho a eketseha ha palo ya dihlopha tsa ethylene glycol e ntse e eketseha.
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Isoleucine CAS: 7004-09-3 Mofani oa Moetsi
Isoleucine (e khutsufalitsoeng e le Ile kapa I) ke amino acid ea α e nang le foromo ea lik'hemik'hale ea HO2CCH(NH2)CH(CH3)CH2CH3. Ke amino acid ea bohlokoa, e bolelang hore batho ba ke ke ba e kopanya, kahoo e tlameha ho metsa. Li-codon tsa eona ke AUU, AUC le AUA. Ka ketane ea lehlakore la hydrocarbon, isoleucine e khetholloa e le amino acid e sa hlokeng hydrophobic. Hammoho le threonine, isoleucine ke e 'ngoe ea li-amino acid tse peli tse tloaelehileng tse nang le ketane ea lehlakore la chiral.
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Arachidonic Acid CAS: 506-32-1 Mofani oa Moetsi
Arachidonic acid (AA, ka linako tse ling ARA) ke mofuta oa omega-6 fatty acid e amehang ho ruruha. Joalo ka li-omega-6 fatty acid tse ling, arachidonic acid e bohlokoa bophelong ba hau. Li-omega-6 fatty acid li thusa ho boloka ts'ebetso ea boko ba hau le ho laola kholo. Ho ja lijo tse nang le motsoako oa omega-6 le omega-3 fatty acids ho tla fokotsa kotsi ea hau ea ho tšoaroa ke lefu la pelo. Arachidonic acid haholo-holo e thusa ho laola ts'ebetso ea methapo.
Phofo ea asiti ea Arachidonic e qhibiliha metsing 'me e bonolo ho e etsa emulsion e tsitsitseng.
