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5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine CAS:733039-20-8
5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine ke motsoako oa lik'hemik'hale o fuputsoang lipatlisisong tsa meriana. E na le sebopeho sa pyrimidine se nang le li-substitution tsa bromo le chloro, tse ka bang bohlokoa bakeng sa lits'ebetso tsa kalafo, tse shebaneng le mekhoa e itseng ea lefu kapa litsela tsa baeloji ho sibolloeng ha meriana.
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4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester CAS:866084-31-3
4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester ke motsoako o rarahaneng oa lik'hemik'hale o nang le mokokotlo oa piperazine o nang le lihlopha tse sebetsang ho kenyeletsoa pyridine, pyrimidine, le tert-butyl ester. Sebopeho sa eona se tšehetsa lits'ebetso tse ka bang teng k'hemistring ea meriana le nts'etsopele ea meriana ka lebaka la mefuta e fapaneng ea pharmacophores.
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Bortezomib CAS:179324-69-7
Bortezomib ke motsoako oa meriana o sebelisoang kalafong ea multiple myeloma le mantle cell lymphoma. Ke oa sehlopha sa li-proteasome inhibitors, tse shebaneng le li-enzyme tsa proteolytic liseleng ho sitisa ts'ebetso ea tsona le ho baka apoptosis (lefu la sele le hlophisitsoeng). Mokhoa ona o etsa hore o sebetse khahlanong le mofetše o itseng moo kholo ea lisele e sa laoleheng e hlahang.
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Methyl 2-bromomethyl-3-nitrobenzoate CAS:98475-07-1
Methyl 2-bromomethyl-3-nitrobenzoate ke motsoako oa lik'hemik'hale o nang le sehlopha sa nitro sebakeng sa 3 le sehlopha sa bromomethyl sebakeng sa 2 sa mokokotlo oa benzoate. E sebelisoa ka har'a motsoako oa lintho tse phelang e le mokhoa o feto-fetohang, o nolofalletsang kaho ea limolek'hule tse rarahaneng tse nang le lihlopha tse itseng tse sebetsang.
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Pemetrexed disodium INT-5 CAS:165049-28-5
Pemetrexed disodium INT-5 ke moriana oa kankere o arotsoeng tlas'a li-antifolate chemotherapy agents. O sebelisoa haholo-holo kalafong ea mefuta e fapaneng ea mofetše, ho kenyeletsoa mesothelioma, mofetše oa matšoafo o seng oa sele e nyane, le mofetše o itseng o metastatic.
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Pemetrexed disodium INT-4 CAS:137281-39-1
Pemetrexed disodium INT-4 ke setlhare sa chemotherapy se thibelang folate se sebediswang ho oncology. E sebediswa kalafong ya mefuta e fapaneng ya kankere, ho kenyeletswa mesothelioma, kankere ya matshwafo e seng ya sele e nyane, le kankere e itseng e melang.
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Pemetrexed disodium INT-3 CAS:155405-80-4
Pemetrexed disodium INT-3 ke setlhare sa chemotherapy se thibelang folate se sebediswang ho oncology. E sebediswa kalafong ya mefuta e fapaneng ya kankere, ho kenyeletswa mesothelioma, kankere ya matshwafo e seng ya sele e nyane, le kankere e itseng e melang.
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Terbinafine botlaaseng CAS:91161-71-6
Terbinafine base ke motsoako o sebetsang oa meriana o sebelisetsoang ho phekola tšoaetso ea fungus. Ke oa sehlopha sa allylamine sa li-antifungal 'me o tsejoa ka katleho ea oona khahlanong le dermatophytes, tomoso le hlobo.
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2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS:3140-73-6
2-Chloro-4,6-dimethoxy-1,3,5-triazine ke motsoako oa lik'hemik'hale o sebelisoang e le motheo oa kaho o feto-fetohang lits'ebetsong tsa tlhahiso ea lintho tse phelang le phetoho ea lik'hemik'hale. E na le lihlopha tse sebetsang tsa chloro le methoxy tse hoketsoeng sebopehong sa lesale la triazine, e nolofalletsang ts'ebeliso ea eona liketsong tse fapaneng tsa lik'hemik'hale le libopeho tsa metsoako.
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2-Amino-4,5-bis(2-methoxyethoxy)benzonitrile CAS:950596-58-4
2-Amino-4,5-bis (2-methoxyethoxy)benzonitrile ke motsoako oa lik'hemik'hale o sebelisoang lipatlisisong tsa meriana, o khetholloang ka sebopeho sa benzonitrile se nang le li-substitution tsa amino le methoxyethoxy, tse ka bang bohlokoa bakeng sa lits'ebetso tse itseng tsa kalafo.
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(1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS:179324-87-9
(1R)-(S)-Pinanediol-1-Ammonium Trifluoroacetate-3-Methylbutane-1-Boronate ke motsoako oa lik'hemik'hale o khetholloang ka sebopeho se rarahaneng se nang le mokokotlo oa pinanediol, sehlopha sa ammonium trifluoroacetate, le ts'ebetso ea boronate ester. E sebelisoa ka har'a motsoako oa lintho tse phelang e le motheo oa chiral, e nolofalletsang ho thehoa ha metsoako e ikhethang le metsoako ea meriana.
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Diethyl L-glutamate hydrochloride CAS:1118-89-4
Diethyl L-glutamate hydrochloride ke motsoako oa lik'hemik'hale o sebelisoang haholo-holo e le motsoako oa maiketsetso lipatlisisong tsa meriana le tlhahiso ea lintho tse phelang. E nkiloe ho L-glutamic acid 'me e sebetsa e le selelekela tlhahisong ea meriana e fapaneng le metsoako e sebetsang ka baeloji.
