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Empagliflozin CAS:864070-44-0 Mofani oa Moetsi

Empagliflozin ke motsoako oa C-glycosyl o nang le masala a beta-glucosyl a nang le sehlopha sa (4-chloro-3-{4-[(3S)-tetrahydrofuran-3-yloxy]benzyl}phenyl setsing sa anomeric. Mothibeli oa sodium-glucose co-transporter 2 o sebelisoang e le tlatsetso lijong le boikoetlisong ho ntlafatsa taolo ea glycemic ho batho ba baholo ba nang le lefu la tsoekere la mofuta oa 2. E na le karolo e le mothibeli oa protheine ea transport ea sodium-glucose subtype 2 le moemeli oa hypoglycemic. Ke motsoako oa C-glycosyl, ether e nkhang hamonate, ether ea tetrahydrofuryl le setho sa monochlorobenzenes.


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Tšebeliso le Phello

Empagliflozin ke sethibela-mafu se secha, se matla le se khethileng sa SGLT-2, se ntlafatsa taolo ea glycemic le litšobotsi tsa metabolic syndrome ho likhoto tse nang le lefu la tsoekere. Empagliflozin (lebitso la khoebo Jardiance) ke sethibela-mafu sa sodium glucose co-transporter-2 (SGLT-2), 'me se etsa hore tsoekere maling e ntšoe ke liphio 'me e ntše ka morotong. Empagliflozin e ka baka ho felloa ke metsi 'meleng' me ea lebisa khatellong e fokotsehileng ea mali, e leng se fellang ka bakuli ba nang le ho tsekela kapa ho akheha le ho fokotseha ha ts'ebetso ea liphio. Kotsi ea bakuli ba hōlileng, haholo-holo ba nang le ts'ebetso e fokolang ea liphio le diuretics, e bonahala e le kholo. FDA e hloka hore Boehring le Eli Lilly ba etse lithuto tse 'ne tsa kamora ho bapatsa: liteko tse felletseng tsa liphello tsa pelo le methapo ea mali tse tsoelang pele, liteko tsa pharmacokinetics ea bana le liteko tsa pharmacodynamics, liteko tsa polokeho le katleho ea bana, teko ea chefo bakeng sa moriana (haholo-holo phello bakeng sa ts'ebetso ea liphio, masapo le kholo le nts'etsopele).

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Ho paka Sehlahisoa:

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Tlhahisoleseling e 'Ngoe:

Sebopeho C23H27ClO7
Teko 99%
Ponahalo Phofo e tšoeu
Nomoro ea CAS 864070-44-0
Ho paka 25KG
Bophelo ba Shelofo lilemo tse 2
Polokelo Boloka sebakeng se pholileng le se omileng
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